We complement our med chem activities with an offer of chemistry solutions for both your drug discovery and development needs
Enantia's support activities include:
Synthesis of cold labelled compounds
Preparation of molecules containing stable isotopes (single to multi-labelled), including deuterated compounds as a strategy to improve pharmacokinetic profile. Exhaustive analysis of synthetic routes and labelled starting materials to design the best route to effectively introduce the required isotopes in the desired positions. Design of positions to be labelled on a case-by-case basis.
Preliminary salt and polymorph screening
The choice of the right solid form of a candidate compound is key to the success of the project. An initial assessment of possible salts and polymorphism is usually carried out at drug discovery stage before performing a full screening study.